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成果及论文

2025年

127. Tianqing Liu; Yuying Li*; Chao Ren; Jianeng Song; Nan Wu; Yan Wang; Zhenghai Huang; Qilei Zhang; Qi Zeng; Jiapei Dai; Xiao-xin Yan; Li Huo*; Mengchao Cui*, The Significant Role of Nitrogen Protonation in the Rational Design of Tau-PET Tracers, ChemRxiv2025, 10.26434/chemrxiv-2025-n82wn.

126. Donglan Huang; Yiming Guo; Mengchao Cui; Hualong Fu*, Development and Preliminary Evaluation of a 125I-Labeled Radioligand ([125I]iodotrazoline) for In Vitro Detection of Imidazoline-2 Binding Site in the Brain, Molecular Pharmaceutics2025, 22(4): 2224-2232.

125. Yimin Chen; Haonan Yu; Wanjia Liu; Ming Wang; Xinlin Wang; Xiaojun Zhang*; Jinming Zhang; Shaobo Yao*; Mengchao Cui*Biphenyl-Trimeric PSMA Theranostic Platform Enables PET Imaging and Optical Detection of Prostate Cancer, Journal of Medicinal Chemistry2025, 68(12): 13075-13088.

124. Yimin Chen; Ming Ni; Xiaojun Zhang; Xinlin Wang; Kaixuan Wang; Qiang Xie*; Jinming Zhang*; Mengchao Cui*Preclinical Evaluation and First-in-Human PET Study of Al18F-Labeled Biphenyl-Based Dimeric PSMA Tracers, Journal of Medicinal Chemistry2025, 68(6): 6832-6843.

123. Fuhai Wu; Xiaoming Wang; Huan Chen; Xu Zhou; Hailong Zhao*Mengchao CuiDevelopment and Validation of an HPLC Method to Determine Chemical and Radiochemical Purity of [18F]Florbetazine Injection, Journal of Labelled Compounds and Radiopharmaceuticals, 2025, 68:e4140.

122. Yue Li; Lili Guan; Xiaoyang Zhang; Jia Li; Xinlin Wang; Wenbo Li; Lu Xu; Shuang Liu; Zhaobing Tang*; Mengchao Cui*; Hua Pang*Dual targeting PET tracer [68Ga]Ga-PSFA-01 in patients with prostate cancers: A pilot exploratory study, Theranostics, 2025, 15(9): 4124-4134.

121. Tianbao Wang; Yufei Qin; Jin-yu Wang; Yihan Xu; Jiaming Guo; Yiling Zhu; Huiyan Zhang; Yujie Qin; Zhong-Quan Qi; Hualong Fu; Ya-jun Liu; Mengchao Cui; Kaixiang Zhou*Less Is More: Donor Engineering of a Stable Molecular Dye for Bioimaging in the NIR-IIb Window, Journal of Medicinal Chemistry2025, 68(3): 3782-3794.

120. Yimin Chen; Wanjia Liu; Ben Li; Xi Gao; Kaixiang Zhou; Mingxin Zhang*; Guangjie Yang*; Mengchao Cui*Synthesis, Preclinical Evaluation, and First-in-Human Assessment of ICG-PSMA-D5: A PSMA-Targeted Probe for Fluorescence-Guided Surgery of Prostate Cancer, Journal of Medicinal Chemistry2025, 68(3): 3858-3872.

119. Xi Gao; Jin-yu Wang; Yufei Qin; Yiling Zhu; Ya-jun Liu; Kaixiang Zhou*; Mengchao Cui*Design, Synthesis, and In Vivo Imaging of a Stable Xanthene-Based Dye with NIR-II Emission up to 1450 nm, Analytical Chemistry2025, 97(3): 1827-1836.

118. Yuqing Xiong; Xinlin Wang; Mengchao Cui*; Yajun Liu*; Beibei Wang*Balancing enthalpy and entropy in inhibitor binding to the prostate-specific membrane antigen (PSMA), Physical Chemistry Chemical Physics2025, 27: 2260-2271.

117. Nan Wu; Xiaojun Zhang; Yuying Li*; Jinming Zhang*; Mengchao Cui*Fluorinated Coumarin Derivatives as Selective PET Tracer for MAO-B Imaging, Journal of Medicinal Chemistry2025, 68(1): 324-337.

116. Xinlin Wang; Xiaoyang Zhang; Xiaojun Zhang; Lili Guan; Xi Gao; Lu Xu; Hua Pang*; Jin Du; Jinming Zhang*Mengchao Cui*; Design, preclinical evaluation, and first-in-human PET study of [68Ga]Ga-PSFA-01: a PSMA/FAP heterobivalent tracer, European Journal of Nuclear Medicine and Molecular Imaging2025, 52: 1166-1176.

115. Tianqing Liu; Chao Ren; Wantong Guo; Xiaojun Zhang; Yuying Li*; Yan Wang; Qilei Zhang; Baian Chen; Jiapei Dai; Xiao-xin Yan; Jinming Zhang; Li Huo*; Mengchao Cui*Synthesis and preclinical evaluation of diarylamine derivative as Tau-PET radiotracer for Alzheimer's Disease, European Journal of Medicinal Chemistry2025, 281: 117046.

2024年

114. Wanqing Li; Xiaojun Zhang; Jie Ma; Jingyin Zhou; Xuan Di; Donglan Huang; Kaixiang Zhou; Jinming Zhang*; Lu Wang*; Hualong Fu*; Mengchao CuiPreclinical Evaluation of Dihydropyrazole-Cored Positron Emission Tomography (PET) Ligands for Imaging of Receptor-Interacting Serine/Threonine Protein Kinase 1 (RIPK1) in the Brain, Journal of Medicinal Chemistry2024, 67(18): 16403-16415.

113. Wanqing Li; Xiaojun Zhang; Jingyin Zhou; Xuan Di; Donglan Huang; Jie Ma; Kaixiang Zhou; Jinming Zhang*; Lu Wang*; Hualong Fu*; Mengchao CuiStructure-based discovery of a 4,5-Dihydropyrazole-cored PET ligand for imaging of receptor-interacting serine/threonine-protein kinase 1 (RIPK1) in the brain, European Journal of Medicinal Chemistry2024, 279: 116803.

112. Jiaming Guo; Yiling Zhu; Yuqian Qu; Longfei Zhang; Mingxi Fang; Zihan Xu; Tianbao Wang; Yufei Qin; Yihan Xu; Yuying Li; Yimin Chen; Hualong Fu; Xiayu Liu; Yajun Liu; Cheng Liu; Yuan Gao; Mengchao Cui; Kaixiang Zhou*Structure Tailoring of Hemicyanine Dyes for In Vivo Shortwave Infrared Imaging, Journal of Medicinal Chemistry2024, 67(18): 16820-16834.

111. Meiqi Wu; Chao Ren; Chenhui Mao; Liling Dong; Bo Li; Xueqian Yang; Zhenghai Huang; Haiqiong Zhang; Yuying Li; Mengshi Yan; Qi Ge; Runze Wu; Feng Feng; Mengchao Cui; Jing Gao; Li Huo*, Evaluation of a novel PET tracer [18F]-Florbetazine for Alzheimer's disease diagnosis and β-amyloid deposition quantification, NeuroImage, 2024, 298, 120779.

110. Ming Ni; Xingxing Zhu; Kaixuan Wang; Wenliang Guo; Qin Shi; Yuying Li; Mengchao Cui*; Qiang Xie*, Novel β-amyloid PET Imaging Study of [18F]92 in Patients with Cognitive Decline, ACS Omega, 2024, 9(32): 34675-34683.

109. Qi Zeng; Xiaojun Zhang; Yuying Li*; Qilei Zhang; Jiapei Dai; Xiao-xin Yan; Yu Liu; Jinming Zhang*; Sen Liu; Mengchao Cui*Discovery and Evaluation of Imidazo[2,1-b][1,3,4]thiadiazole Derivatives as New Candidates for α-Synuclein PET Imaging, Journal of Medicinal Chemistry2024, 67(15): 12695-12710.

108. Xiaohui Luan; Shaoxi Niu; Yachao Liu; Xiaojun Zhang; Xiaodan Xu; Shuwei Sun; Yabing Sun; Jingfeng Zhang; Yuan Wang; Zhiqiang Chen; Yimin Chen; Mengchao Cui; Ruimin Wang; Xu Zhang*; Jinming Zhang*; Baixuan Xu*. The first-in-human preclinical evaluation of the new probe [123I]I-PSMA-7 for real-time intraoperative targeted biopsy and SPECT/CT imaging in prostate cancer, European Journal of Nuclear Medicine and Molecular Imaging2024, 51: 4141-4150.

107. Yuying Li; Xiaojun Zhang; Hailong Zhao; Yan Wang; Dandan Zhang; Xiaoming Wang; Ruilin Dong; Xiao-xin Yan; Jing Wu; Yanying Sui; Jinming Zhang*; Mengchao Cui*Screening of [18F]Florbetazine for Aβ Plaques and a Head-to-Head Comparison Study with [11C]Pittsburgh Compound-B ([11C]PiB) in Human SubjectsACS Pharmacology & Translational Science, 2024, 7(7): 2054-2062.

106. Cao Lu; Cong Meng; Yuying Li; Jinling Yuan; Xiaojun Ren; Liang Gao; Dongdong Su; Kai Cao; Mengchao Cui; Qing Yuan*; Xueyun Gao*, A probe for NIR-II imaging and multimodal analysis of early Alzheimer’s disease by targeting CTGFNature Communications, 2024, 48(3): 166-177.

105. Wantong Guo; Yuying Li; Mengchao Cui*Research Progress of PET Imaging Agents Targeting Abnormal Protein Aggregates in the BrainProgress in Pharmaceutical Sciences, 2024, 48(3): 166-177. 

104. Qi-Jie Zhang; Jie Lin; You-Liang Wang; Long Chen; Ying Ding; Fu-Ze Zheng; Huan-Huan Song; Ao-Wei Lv; Yu-Ying Li; Qi-Fu Guo; Min-Ting Lin; Wei Hu; Liu-Qing Xu; Wen-Long Zhao; Ling Fang; Meng-Chao Cui; Zhi-Fei Fu; Wan-Jin Chen; Jing Zhang*; Zhi-Qiang Wang*; Ning Wang*; Ying Fu*Detection of pTDP-43 via routine muscle biopsy: A promising diagnostic biomarker for amyotrophic lateral sclerosis, Brain Pathology, 2024, e13261.

103. Yuying Li; Tianqing Liu; Qi Zeng; Mengchao Cui*Current status of PET tracers for the early diagnosis of Alzheimer's diseaseTrAC Trends in Analytical Chemistry, 2024, 172(10284):117546.

2023年

102. Longfei Zhang; Xiaojing Shi; Yuying Li; Xiaojiang Duan; Xing Yang; Zhenhua Hu*; Mengchao Cui*, An NIR-II Probe with High PSMA Affinity Demonstrates an Unexpected Excellent Bone Imaging Ability, Journal of Medicinal Chemistry2023, 66, 23, 16441-16454.